Azastene

Azastene is a synthetic anabolic-androgenic steroid (AAS). It is derived from dihydrotestosterone (DHT) and possesses a 17α-methyl group, which allows for oral administration. Azastene is primarily known for its use in research settings and has not been widely marketed or approved for human use in most countries.

Pharmacology

Azastene functions as an androgen receptor agonist, similar to other AAS. It binds to the androgen receptor, which leads to increased protein synthesis, nitrogen retention, and muscle growth. The 17α-methylation contributes to its oral bioavailability but also potentially increases its hepatotoxicity.

Effects and Uses

While not widely studied or clinically used, the intended effects of azastene, based on its structural similarity to other AAS, would likely include:

• Increased muscle mass
• Increased strength
• Reduced body fat
• Increased bone density

These effects, however, are accompanied by a range of potential side effects.

Side Effects

As with other AAS, azastene carries a risk of significant side effects, including:

• Liver damage (hepatotoxicity) due to the 17α-methylation
• Cardiovascular issues, such as increased cholesterol levels and blood pressure
• Suppression of natural testosterone production
• Acne
• Hair loss
• Gynecomastia (breast enlargement in males)
• Virilization (development of male characteristics in females)

Legal Status

Azastene is generally not approved for human use in most countries and may be considered a controlled substance or prohibited for use in sports. Its legal status varies depending on the specific jurisdiction.

Disclaimer: This information is for educational purposes only and should not be considered medical advice. The use of anabolic-androgenic steroids carries significant health risks and is often illegal. Consult with a qualified healthcare professional before making any decisions related to your health or treatment.